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-Structure paper
Title | New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 1492-1500, Year 2016 |
Publish date | Aug 26, 2015 (structure data deposition date) |
Authors | Baud, M.G. / Lin-Shiao, E. / Zengerle, M. / Tallant, C. / Ciulli, A. |
External links | J. Med. Chem. / PubMed:26367539 |
Methods | X-ray diffraction |
Resolution | 1.4 - 1.5 Å |
Structure data | PDB-5dfb: PDB-5dfc: PDB-5dfd: |
Chemicals | ChemComp-NI: ChemComp-2PE: ChemComp-GOL: ChemComp-HOH: ChemComp-EAM: ChemComp-59E: |
Source |
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Keywords | TRANSCRIPTION / Transcription factors / BET bromodomains / protein mutation engineering / molecular probes |