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-Structure paper
Title | New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 1492-1500, Year 2016 |
Publish date | Aug 26, 2015 (structure data deposition date) |
![]() | Baud, M.G. / Lin-Shiao, E. / Zengerle, M. / Tallant, C. / Ciulli, A. |
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Methods | X-ray diffraction |
Resolution | 1.4 - 1.5 Å |
Structure data | ![]() PDB-5dfb: ![]() PDB-5dfc: ![]() PDB-5dfd: |
Chemicals | ![]() ChemComp-NI: ![]() ChemComp-2PE: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-EAM: ![]() ChemComp-59E: |
Source |
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![]() | TRANSCRIPTION / Transcription factors / BET bromodomains / protein mutation engineering / molecular probes |