+Search query
-Structure paper
Title | Identification and Characterization of an Irreversible Inhibitor of CDK2. |
---|---|
Journal, issue, pages | Chem. Biol., Vol. 22, Page 1159-1164, Year 2015 |
Publish date | Jul 30, 2015 (structure data deposition date) |
Authors | Anscombe, E. / Meschini, E. / Mora-Vidal, R. / Martin, M.P. / Staunton, D. / Geitmann, M. / Danielson, U.H. / Stanley, W.A. / Wang, L.Z. / Reuillon, T. ...Anscombe, E. / Meschini, E. / Mora-Vidal, R. / Martin, M.P. / Staunton, D. / Geitmann, M. / Danielson, U.H. / Stanley, W.A. / Wang, L.Z. / Reuillon, T. / Golding, B.T. / Cano, C. / Newell, D.R. / Noble, M.E. / Wedge, S.R. / Endicott, J.A. / Griffin, R.J. |
External links | Chem. Biol. / PubMed:26320860 |
Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | PDB-5cyi: |
Chemicals | ChemComp-55S: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE / CDK2 Cyclin A covalent inhibitor vinylsulphone |