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-Structure paper
Title | BGB-283, a Novel RAF Kinase and EGFR Inhibitor, Displays Potent Antitumor Activity in BRAF-Mutated Colorectal Cancers. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 14, Page 2187-2197, Year 2015 |
Publish date | Aug 22, 2014 (structure data deposition date) |
![]() | Tang, Z. / Yuan, X. / Du, R. / Cheung, S.H. / Zhang, G. / Wei, J. / Zhao, Y. / Feng, Y. / Peng, H. / Zhang, Y. ...Tang, Z. / Yuan, X. / Du, R. / Cheung, S.H. / Zhang, G. / Wei, J. / Zhao, Y. / Feng, Y. / Peng, H. / Zhang, Y. / Du, Y. / Hu, X. / Gong, W. / Liu, Y. / Gao, Y. / Hao, R. / Li, S. / Wang, S. / Ji, J. / Zhang, L. / Sutton, D. / Wei, M. / Zhou, C. / Wang, L. / Luo, L. |
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Methods | X-ray diffraction |
Resolution | 3.5 Å |
Structure data | ![]() PDB-4r5y: |
Chemicals | ![]() ChemComp-3K3: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / signal transduction / TRANSFERASE-TRANSFERASE INHIBITOR complex |