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-Structure paper
Title | Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 1340-1349, Year 2016 |
Publish date | Jun 11, 2014 (structure data deposition date) |
![]() | Xu, M. / Unzue, A. / Dong, J. / Spiliotopoulos, D. / Nevado, C. / Caflisch, A. |
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Methods | X-ray diffraction |
Resolution | 1.7 Å |
Structure data | ![]() PDB-4tqn: |
Chemicals | ![]() ChemComp-UL4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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