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-Structure paper
Title | Structure-based development of nitroxoline derivatives as potential multifunctional anti-Alzheimer agents. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 23, Page 4442-4452, Year 2015 |
Publish date | Jan 7, 2015 (structure data deposition date) |
Authors | Knez, D. / Brus, B. / Coquelle, N. / Sosic, I. / Sink, R. / Brazzolotto, X. / Mravljak, J. / Colletier, J.P. / Gobec, S. |
External links | Bioorg. Med. Chem. / PubMed:26116179 |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | PDB-4xii: |
Chemicals | ChemComp-40V: ChemComp-NAG: ChemComp-FUL: ChemComp-FUC: ChemComp-CL: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / anti-alzherimer / huBuche / human butyrylcholinesterase / metal chelator / abeta peptide / ab aggregation |