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-Structure paper
Title | Fragment-Based Discovery of a Small Molecule Inhibitor of Bruton's Tyrosine Kinase. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 5437-5444, Year 2015 |
Publish date | Mar 31, 2015 (structure data deposition date) |
Authors | Smith, C.R. / Dougan, D.R. / Komandla, M. / Kanouni, T. / Knight, B. / Lawson, J.D. / Sabat, M. / Taylor, E.R. / Vu, P. / Wyrick, C. |
External links | J. Med. Chem. / PubMed:26087137 |
Methods | X-ray diffraction |
Resolution | 1.6 - 2 Å |
Structure data | PDB-4z3v: PDB-4zly: PDB-4zlz: |
Chemicals | ChemComp-IMD: ChemComp-IPA: ChemComp-EDO: ChemComp-4L6: ChemComp-HOH: ChemComp-DMS: ChemComp-4RU: ChemComp-4RV: |
Source |
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Keywords | TRANSFERASE / cytoplasmic tyrosine kinase / transcriptional regulation / nuclear factor-kappaB / Transferase/Transferase Inhibitor / Transferase-Transferase Inhibitor complex |