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-Structure paper
Title | Structure-Based Design of gamma-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 4927-4939, Year 2015 |
Publish date | Apr 9, 2015 (structure data deposition date) |
![]() | Ran, X. / Zhao, Y. / Liu, L. / Bai, L. / Yang, C.Y. / Zhou, B. / Meagher, J.L. / Chinnaswamy, K. / Stuckey, J.A. / Wang, S. |
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Methods | X-ray diffraction |
Resolution | 1.27 Å |
Structure data | ![]() PDB-4z93: |
Chemicals | ![]() ChemComp-4LD: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / Bromodomain |