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-Structure paper
Title | Peroxisome proliferator-activated receptor gamma (PPAR gamma ) has multiple binding points that accommodate ligands in various conformations: Structurally similar PPAR gamma partial agonists bind to PPAR gamma LBD in different conformations |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 25, Page 2758-2762, Year 2015 |
Publish date | Mar 17, 2015 (structure data deposition date) |
Authors | Ohashi, M. / Gamo, K. / Oyama, T. / Miyachi, H. |
External links | Bioorg. Med. Chem. Lett. / PubMed:26025876 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-4yt1: |
Chemicals | ChemComp-JJB: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / NUCLEAR RECEPTOR |