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-Structure paper
Title | Discovery of a new chemical series of BRD4(1) inhibitors using protein-ligand docking and structure-guided design. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 25, Page 2818-2823, Year 2015 |
Publish date | Feb 26, 2015 (structure data deposition date) |
![]() | Duffy, B.C. / Liu, S. / Martin, G.S. / Wang, R. / Hsia, M.M. / Zhao, H. / Guo, C. / Ellis, M. / Quinn, J.F. / Kharenko, O.A. ...Duffy, B.C. / Liu, S. / Martin, G.S. / Wang, R. / Hsia, M.M. / Zhao, H. / Guo, C. / Ellis, M. / Quinn, J.F. / Kharenko, O.A. / Norek, K. / Gesner, E.M. / Young, P.R. / McLure, K.G. / Wagner, G.S. / Lakshminarasimhan, D. / White, A. / Suto, R.K. / Hansen, H.C. / Kitchen, D.B. |
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Methods | X-ray diffraction |
Resolution | 1.33 - 1.6 Å |
Structure data | ![]() PDB-4yh3: ![]() PDB-4yh4: |
Chemicals | ![]() ChemComp-Y80: ![]() ChemComp-HOH: ![]() ChemComp-Y81: ![]() ChemComp-GOL: ![]() ChemComp-NA: |
Source |
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