+Search query
-Structure paper
Title | Evolution and synthesis of novel orally bioavailable inhibitors of PDE10A. |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 25, Page 1864-1868, Year 2015 |
Publish date | Mar 13, 2015 (structure data deposition date) |
![]() | Burdi, D.F. / Campbell, J.E. / Wang, J. / Zhao, S. / Zhong, H. / Wei, J. / Campbell, U. / Shao, L. / Herman, L. / Koch, P. ...Burdi, D.F. / Campbell, J.E. / Wang, J. / Zhao, S. / Zhong, H. / Wei, J. / Campbell, U. / Shao, L. / Herman, L. / Koch, P. / Jones, P.G. / Hewitt, M.C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.308 - 2.502 Å |
Structure data | ![]() PDB-4yqh: ![]() PDB-4ys7: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-4F7: ![]() ChemComp-HOH: ![]() ChemComp-4GK: |
Source |
|
![]() | HYDROLASE/HYDROLASE INHIBITOR / inhibitor / PDE10A / co-crystal / HYDROLASE-HYDROLASE INHIBITOR complex |