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Title | Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 4080-4085, Year 2015 |
Publish date | Mar 4, 2015 (structure data deposition date) |
Authors | Hoang, H.N. / Song, K. / Hill, T.A. / Derksen, D.R. / Edmonds, D.J. / Kok, W.M. / Limberakis, C. / Liras, S. / Loria, P.M. / Mascitti, V. ...Hoang, H.N. / Song, K. / Hill, T.A. / Derksen, D.R. / Edmonds, D.J. / Kok, W.M. / Limberakis, C. / Liras, S. / Loria, P.M. / Mascitti, V. / Mathiowetz, A.M. / Mitchell, J.M. / Piotrowski, D.W. / Price, D.A. / Stanton, R.V. / Suen, J.Y. / Withka, J.M. / Griffith, D.A. / Fairlie, D.P. |
External links | J. Med. Chem. / PubMed:25839426 |
Methods | NMR (solution) |
Structure data | PDB-2n08: PDB-2n09: PDB-2n0i: PDB-2n0n: |
Keywords | DE NOVO PROTEIN / hydrophobic peptide / GLP-1R agonist |