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-Structure paper
Title | Discovery of Novel P1 Groups for Coagulation Factor VIIa Inhibition Using Fragment-Based Screening. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 2799-2808, Year 2015 |
Publish date | Dec 10, 2014 (structure data deposition date) |
![]() | Cheney, D.L. / Bozarth, J.M. / Metzler, W.J. / Morin, P.E. / Mueller, L. / Newitt, J.A. / Nirschl, A.H. / Rendina, A.R. / Tamura, J.K. / Wei, A. ...Cheney, D.L. / Bozarth, J.M. / Metzler, W.J. / Morin, P.E. / Mueller, L. / Newitt, J.A. / Nirschl, A.H. / Rendina, A.R. / Tamura, J.K. / Wei, A. / Wen, X. / Wurtz, N.R. / Seiffert, D.A. / Wexler, R.R. / Priestley, E.S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.5 Å |
Structure data | ![]() PDB-4x8s: ![]() PDB-4x8t: ![]() PDB-4x8u: ![]() PDB-4x8v: |
Chemicals | ![]() ChemComp-3Z7: ![]() ChemComp-CA: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-3Z8: ![]() ChemComp-3ZB: ![]() ChemComp-3Z9: |
Source |
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![]() | hydrolase/hydrolase inhibitor / GLYCOPROTEIN / HYDROLASE / SERINE PROTEASE / PLASMA / BLOOD COAGULATION FACTOR / PROTEIN INHIBITOR COMPLEX / CALCIUM- BINDING / hydrolase-hydrolase inhibitor complex |