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Title | A Potent, Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3). |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 54, Page 5166-5170, Year 2015 |
Publish date | Dec 15, 2014 (structure data deposition date) |
Authors | Kaniskan, H.U. / Szewczyk, M.M. / Yu, Z. / Eram, M.S. / Yang, X. / Schmidt, K. / Luo, X. / Dai, M. / He, F. / Zang, I. ...Kaniskan, H.U. / Szewczyk, M.M. / Yu, Z. / Eram, M.S. / Yang, X. / Schmidt, K. / Luo, X. / Dai, M. / He, F. / Zang, I. / Lin, Y. / Kennedy, S. / Li, F. / Dobrovetsky, E. / Dong, A. / Smil, D. / Min, S.J. / Landon, M. / Lin-Jones, J. / Huang, X.P. / Roth, B.L. / Schapira, M. / Atadja, P. / Barsyte-Lovejoy, D. / Arrowsmith, C.H. / Brown, P.J. / Zhao, K. / Jin, J. / Vedadi, M. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:25728001 |
Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | PDB-4ryl: |
Chemicals | ChemComp-3ZG: ChemComp-UNX: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / PRMT3 / SGC707 / Structural Genomics / Structural Genomics Consortium |