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Title | Structure Enabled Design of BAZ2-ICR, A Chemical Probe Targeting the Bromodomains of BAZ2A and BAZ2B. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 2553-2559, Year 2015 |
Publish date | Jan 25, 2015 (structure data deposition date) |
![]() | Drouin, L. / McGrath, S. / Vidler, L.R. / Chaikuad, A. / Monteiro, O. / Tallant, C. / Philpott, M. / Rogers, C. / Fedorov, O. / Liu, M. ...Drouin, L. / McGrath, S. / Vidler, L.R. / Chaikuad, A. / Monteiro, O. / Tallant, C. / Philpott, M. / Rogers, C. / Fedorov, O. / Liu, M. / Akhtar, W. / Hayes, A. / Raynaud, F. / Muller, S. / Knapp, S. / Hoelder, S. |
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Methods | X-ray diffraction |
Resolution | 1.75 - 1.98 Å |
Structure data | ![]() PDB-4xua: ![]() PDB-4xub: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-43C: ![]() ChemComp-HOH: ![]() ChemComp-43D: |
Source |
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![]() | TRANSCRIPTION / bromodomain / acetylated lysine binding protein / KIAA1476 / WALp4 / Structural Genomics / Structural Genomics Consortium / SGC |