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-Structure paper
Title | Distinct binding mode of multikinase inhibitor lenvatinib revealed by biochemical characterization. |
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Journal, issue, pages | ACS MED. CHEM. LETT., Vol. 6, Page 89-94, Year 2015 |
Publish date | Sep 24, 2014 (structure data deposition date) |
![]() | Okamoto, K. / Ikemori-Kawada, M. / Jestel, A. / von Konig, K. / Funahashi, Y. / Matsushima, T. / Tsuruoka, A. / Inoue, A. / Matsui, J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.57 - 1.9 Å |
Structure data | ![]() PDB-3wzd: ![]() PDB-3wze: |
Chemicals | ![]() ChemComp-LEV: ![]() ChemComp-DTT: ![]() ChemComp-EDO: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-BAX: ![]() ChemComp-ACT: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / KDR RECEPTOR KINASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |