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-Structure paper
Title | Structure-Based Drug Design of Novel Potent and Selective Tetrahydropyrazolo[1,5-a]pyrazines as ATR Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 37-41, Year 2015 |
Publish date | Aug 29, 2014 (structure data deposition date) |
![]() | Barsanti, P.A. / Aversa, R.J. / Jin, X. / Pan, Y. / Lu, Y. / Elling, R. / Jain, R. / Knapp, M. / Lan, J. / Lin, X. ...Barsanti, P.A. / Aversa, R.J. / Jin, X. / Pan, Y. / Lu, Y. / Elling, R. / Jain, R. / Knapp, M. / Lan, J. / Lin, X. / Rudewicz, P. / Sim, J. / Taricani, L. / Thomas, G. / Xiao, L. / Yue, Q. |
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Methods | X-ray diffraction |
Resolution | 2.39 Å |
Structure data | ![]() PDB-4waf: |
Chemicals | ![]() ChemComp-3K6: ![]() ChemComp-HOH: |
Source |
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![]() | transferase/transferase inhibitor / PI3K / chimera / lipid kinase / transferase-transferase inhibitor complex |