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| Title | Direct inhibitors of InhA are active against Mycobacterium tuberculosis |
|---|---|
| Journal, issue, pages | Sci Transl Med, Vol. 7, Page 269ra3-269ra3, Year 2015 |
| Publish date | Sep 7, 2014 (structure data deposition date) |
Authors | Manjunatha, U.H. / Rao, S.P.S. / Kondreddi, R.R. / Noble, C.G. / Camacho, L.R. / Tan, B.H. / Ng, S.H. / Ng, P.S. / Ma, N.L. / Lakshminarayana, S.B. ...Manjunatha, U.H. / Rao, S.P.S. / Kondreddi, R.R. / Noble, C.G. / Camacho, L.R. / Tan, B.H. / Ng, S.H. / Ng, P.S. / Ma, N.L. / Lakshminarayana, S.B. / Herve, M. / Barnes, S.W. / Yu, W. / Kuhen, K. / Blasco, F. / Beer, D. / Walker, J.R. / Tonge, P.J. / Glynne, R. / Smith, P.W. / Diagana, T.T. |
External links | Sci Transl Med / PubMed:25568071 |
| Methods | X-ray diffraction |
| Resolution | 2.9 - 3.2 Å |
| Structure data | ![]() PDB-4r9r: ![]() PDB-4r9s: |
| Chemicals | ![]() ChemComp-NAD: ![]() ChemComp-3KX: ![]() ChemComp-HOH: ![]() ChemComp-3KY: |
| Source |
|
Keywords | OXIDOREDUCTASE / enoyl-acyl carrier protein reductase / enoyl acyl carrier protein reductase |
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mycobacterium tuberculosis h37rv (bacteria)
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