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-Structure paper
Title | Tricyclic Covalent Inhibitors Selectively Target Jak3 through an Active Site Thiol. |
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Journal, issue, pages | J. Biol. Chem., Vol. 290, Page 4573-4589, Year 2015 |
Publish date | Jun 24, 2014 (structure data deposition date) |
![]() | Goedken, E.R. / Argiriadi, M.A. / Banach, D.L. / Fiamengo, B.A. / Foley, S.E. / Frank, K.E. / George, J.S. / Harris, C.M. / Hobson, A.D. / Ihle, D.C. ...Goedken, E.R. / Argiriadi, M.A. / Banach, D.L. / Fiamengo, B.A. / Foley, S.E. / Frank, K.E. / George, J.S. / Harris, C.M. / Hobson, A.D. / Ihle, D.C. / Marcotte, D. / Merta, P.J. / Michalak, M.E. / Murdock, S.E. / Tomlinson, M.J. / Voss, J.W. |
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Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-4qps: |
Chemicals | ![]() ChemComp-37Q: ![]() ChemComp-HOH: |
Source |
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![]() | Transferase/transferase inhibitor / Kinase catalytic domain / TRANSFERASE / Transferase-transferase inhibitor complex |