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-Structure paper
Title | A new class of peptidomimetics targeting the polo-box domain of polo-like kinase 1. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 294-304, Year 2015 |
Publish date | Sep 16, 2014 (structure data deposition date) |
Authors | Ahn, M. / Han, Y.H. / Park, J.E. / Kim, S. / Lee, W.C. / Lee, S.J. / Gunasekaran, P. / Cheong, C. / Shin, S.Y. / Kim, H.Y. ...Ahn, M. / Han, Y.H. / Park, J.E. / Kim, S. / Lee, W.C. / Lee, S.J. / Gunasekaran, P. / Cheong, C. / Shin, S.Y. / Kim, H.Y. / Ryu, E.K. / Murugan, R.N. / Kim, N.H. / Bang, J.K. |
External links | J. Med. Chem. / PubMed:25347203 |
Methods | X-ray diffraction |
Resolution | 1.6 - 2.71 Å |
Structure data | PDB-4rcp: PDB-4whh: PDB-4whk: PDB-4whl: |
Chemicals | ChemComp-EDO: ChemComp-HOH: ChemComp-SO4: |
Source |
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Keywords | Transferase/transferase inhibitor / Polo-box domain / Transferase-transferase inhibitor complex / Polo-like kinase / inhibitor / peptide derivative |