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-Structure paper
Title | Discovery of Novel, Dual Mechanism ERK Inhibitors by Affinity Selection Screening of an Inactive Kinase. |
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Journal, issue, pages | J. Med. Chem., Vol. 57, Page 8817-8826, Year 2014 |
Publish date | Jul 26, 2014 (structure data deposition date) |
![]() | Deng, Y. / Shipps, G.W. / Cooper, A. / English, J.M. / Annis, D.A. / Carr, D. / Nan, Y. / Wang, T. / Zhu, H.Y. / Chuang, C.C. ...Deng, Y. / Shipps, G.W. / Cooper, A. / English, J.M. / Annis, D.A. / Carr, D. / Nan, Y. / Wang, T. / Zhu, H.Y. / Chuang, C.C. / Dayananth, P. / Hruza, A.W. / Xiao, L. / Jin, W. / Kirschmeier, P. / Windsor, W.T. / Samatar, A.A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.65 Å |
Structure data | ![]() PDB-4qyy: |
Chemicals | ![]() ChemComp-3G7: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE / SERINE/THREONINE-PROTEIN KINASE / MAP KINASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |