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-Structure paper
Title | Novel human D-amino acid oxidase inhibitors stabilize an active-site lid-open conformation. |
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Journal, issue, pages | Biosci. Rep., Vol. 34, Year 2014 |
Publish date | May 20, 2014 (structure data deposition date) |
![]() | Terry-Lorenzo, R.T. / Chun, L.E. / Brown, S.P. / Heffernan, M.L. / Fang, Q.K. / Orsini, M.A. / Pollegioni, L. / Hardy, L.W. / Spear, K.L. / Large, T.H. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 - 2.85 Å |
Structure data | ![]() PDB-4qfc: ![]() PDB-4qfd: |
Chemicals | ![]() ChemComp-FAD: ![]() ChemComp-31T: ![]() ChemComp-K: ![]() ChemComp-HOH: ![]() ChemComp-NA: ![]() ChemComp-31R: |
Source |
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![]() | oxidoreductase/oxidoreductase inhibitor / OXIDASE / OXIDOREDUCTASE / DAAO / D-AMINO ACID OXIDASE / FAD dependent / NMDAR / schizophrenia / D-serine competitive / oxidoreductase-oxidoreductase inhibitor complex / NMDA receptor |