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-Structure paper
Title | Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 22, Page 4099-4108, Year 2014 |
Publish date | Nov 2, 2013 (structure data deposition date) |
![]() | Tykvart, J. / Schimer, J. / Barinkova, J. / Pachl, P. / Postova-Slavetinska, L. / Majer, P. / Konvalinka, J. / Sacha, P. |
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Methods | X-ray diffraction |
Resolution | 1.63 - 2.31 Å |
Structure data | ![]() PDB-4ngm: ![]() PDB-4ngn: ![]() PDB-4ngp: ![]() PDB-4ngq: ![]() PDB-4ngr: ![]() PDB-4ngs: ![]() PDB-4ngt: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-ZN: ![]() ChemComp-CL: ![]() ChemComp-CA: ![]() ChemComp-JB7: ![]() ChemComp-HOH: ![]() ChemComp-J96: ![]() ChemComp-J31: ![]() ChemComp-J37: ![]() ChemComp-J21: ![]() ChemComp-J34: ![]() ChemComp-NA: ![]() ChemComp-J42: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / hydrolase / glutamate carboxypeptidase II / PSMA / NAALADASE / urea-based inhibitor / caboxypeptidase / glycoprotein / metallopeptidase / HYDROLASE-HYDROLASE INHIBITOR complex / trasmembrane |