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-Structure paper
Title | Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 4, Page 353-357, Year 2013 |
Publish date | Dec 6, 2012 (structure data deposition date) |
Authors | Bolshan, Y. / Getlik, M. / Kuznetsova, E. / Wasney, G.A. / Hajian, T. / Poda, G. / Nguyen, K.T. / Wu, H. / Dombrovski, L. / Dong, A. ...Bolshan, Y. / Getlik, M. / Kuznetsova, E. / Wasney, G.A. / Hajian, T. / Poda, G. / Nguyen, K.T. / Wu, H. / Dombrovski, L. / Dong, A. / Senisterra, G. / Schapira, M. / Arrowsmith, C.H. / Brown, P.J. / Al-Awar, R. / Vedadi, M. / Smil, D. |
External links | ACS Med Chem Lett / PubMed:24900672 |
Methods | X-ray diffraction |
Resolution | 1.66 Å |
Structure data | PDB-4ia9: |
Chemicals | ChemComp-IA9: ChemComp-EDO: ChemComp-UNX: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / WDR5 / STRUCTURAL GENOMICS CONSORTIUM / WD REPEAT DOMAIN 5 / SGC |