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-Structure paper
Title | Identification of an Adamantyl Azaquinolone JNK Selective Inhibitor. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 3, Page 764-768, Year 2012 |
Publish date | Mar 16, 2012 (structure data deposition date) |
Authors | Haynes, N.E. / Scott, N.R. / Chen, L.C. / Janson, C.A. / Li, J.K. / Lukacs, C.M. / Railkar, A. / Tozzo, E. / Whittard, T. / Brown, N.F. / Cheung, A.W. |
External links | ACS Med Chem Lett / PubMed:24900545 |
Methods | X-ray diffraction |
Resolution | 2.27 Å |
Structure data | PDB-4e73: |
Chemicals | ChemComp-0NR: ChemComp-HOH: |
Source |
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Keywords | Transferase/Transferase Inhibitor / Kinase / Transferase-Transferase Inhibitor complex |