+Search query
-Structure paper
Title | Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization. |
---|---|
Journal, issue, pages | ACS Med Chem Lett, Vol. 3, Page 278-283, Year 2012 |
Publish date | Oct 10, 2011 (structure data deposition date) |
![]() | Dowling, J.E. / Chuaqui, C. / Pontz, T.W. / Lyne, P.D. / Larsen, N.A. / Block, M.H. / Chen, H. / Su, N. / Wu, A. / Russell, D. ...Dowling, J.E. / Chuaqui, C. / Pontz, T.W. / Lyne, P.D. / Larsen, N.A. / Block, M.H. / Chen, H. / Su, N. / Wu, A. / Russell, D. / Pollard, H. / Lee, J.W. / Peng, B. / Thakur, K. / Ye, Q. / Zhang, T. / Brassil, P. / Racicot, V. / Bao, L. / Denz, C.R. / Cooke, E. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-3u4u: |
Chemicals | ![]() ChemComp-LNH: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
|
![]() | Transferase/Transferase Inhibitor / Kinase / Transferase / Inhibitor binding / Transferase-Transferase Inhibitor complex |