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-Structure paper
Title | Discovery of GNF-5837, a Selective TRK Inhibitor with Efficacy in Rodent Cancer Tumor Models. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 3, Page 140-145, Year 2012 |
Publish date | Dec 16, 2011 (structure data deposition date) |
![]() | Albaugh, P. / Fan, Y. / Mi, Y. / Sun, F. / Adrian, F. / Li, N. / Jia, Y. / Sarkisova, Y. / Kreusch, A. / Hood, T. ...Albaugh, P. / Fan, Y. / Mi, Y. / Sun, F. / Adrian, F. / Li, N. / Jia, Y. / Sarkisova, Y. / Kreusch, A. / Hood, T. / Lu, M. / Liu, G. / Huang, S. / Liu, Z. / Loren, J. / Tuntland, T. / Karanewsky, D.S. / Seidel, H.M. / Molteni, V. |
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Methods | X-ray diffraction |
Resolution | 2.2001 Å |
Structure data | ![]() PDB-3v5q: |
Chemicals | ![]() ChemComp-CL: ![]() ChemComp-0F4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / ![]() ![]() ![]() |