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-Structure paper
Title | 2-Amino-7-substituted benzoxazole analogs as potent RSK2 inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 24, Page 1592-1596, Year 2014 |
Publish date | Dec 5, 2013 (structure data deposition date) |
Authors | Costales, A. / Mathur, M. / Ramurthy, S. / Lan, J. / Subramanian, S. / Jain, R. / Atallah, G. / Setti, L. / Lindvall, M. / Appleton, B.A. ...Costales, A. / Mathur, M. / Ramurthy, S. / Lan, J. / Subramanian, S. / Jain, R. / Atallah, G. / Setti, L. / Lindvall, M. / Appleton, B.A. / Ornelas, E. / Feucht, P. / Warne, B. / Doyle, L. / Basham, S.E. / Aronchik, I. / Jefferson, A.B. / Shafer, C.M. |
External links | Bioorg. Med. Chem. Lett. / PubMed:24534486 |
Methods | X-ray diffraction |
Resolution | 1.74 - 1.94 Å |
Structure data | PDB-4nw5: PDB-4nw6: |
Chemicals | ChemComp-2NR: ChemComp-HOH: ChemComp-2NS: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |