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-Structure paper
Title | The identification of AF38469: An orally bioavailable inhibitor of the VPS10P family sorting receptor Sortilin. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 24, Page 177-180, Year 2014 |
Publish date | Oct 15, 2013 (structure data deposition date) |
![]() | Schrder, T.J. / Christensen, S. / Lindberg, S. / Langgard, M. / David, L. / Maltas, P.J. / Eskildsen, J. / Jacobsen, J. / Tagmose, L. / Simonsen, K.B. ...Schrder, T.J. / Christensen, S. / Lindberg, S. / Langgard, M. / David, L. / Maltas, P.J. / Eskildsen, J. / Jacobsen, J. / Tagmose, L. / Simonsen, K.B. / Biilmann Rnn, L.C. / de Jong, I.E. / Malik, I.J. / Karlsson, J.J. / Bundgaard, C. / Egebjerg, J. / Stavenhagen, J.B. / Strandbygard, D. / Thirup, S. / Andersen, J.L. / Uppalanchi, S. / Pervaram, S. / Kasturi, S.P. / Eradi, P. / Sakumudi, D.R. / Watson, S.P. |
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Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-4n7e: |
Chemicals | ![]() ChemComp-PGE: ![]() ChemComp-2JQ: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN / Sortilin / Small molecule ligand / AF38469 / AF40431 / proNGF / Alzheimer's disease / Beta-propeller Asp-box repeat / Vps10p domain / 10CC domain / Receptor Sorting / Membrane |