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Title | Rationally designed inhibitor targeting antigen-trimming aminopeptidases enhances antigen presentation and cytotoxic T-cell responses. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 110, Page 19890-19895, Year 2013 |
Publish date | Feb 20, 2013 (structure data deposition date) |
![]() | Zervoudi, E. / Saridakis, E. / Birtley, J.R. / Seregin, S.S. / Reeves, E. / Kokkala, P. / Aldhamen, Y.A. / Amalfitano, A. / Mavridis, I.M. / James, E. ...Zervoudi, E. / Saridakis, E. / Birtley, J.R. / Seregin, S.S. / Reeves, E. / Kokkala, P. / Aldhamen, Y.A. / Amalfitano, A. / Mavridis, I.M. / James, E. / Georgiadis, D. / Stratikos, E. |
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Methods | X-ray diffraction |
Resolution | 2.789 Å |
Structure data | ![]() PDB-4jbs: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-ZN: ![]() ChemComp-P52: ![]() ChemComp-IMD: ![]() ChemComp-HOH: |
Source |
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![]() | Hydrolase/Hydrolase Inhibitor / Thermolysin-like catalytic domain / Hydrolase / Aminopeptidase / Zinc binding / Endoplasmic Reticulum / Hydrolase-Hydrolase Inhibitor complex |