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-Structure paper
Title | Staurosporine-derived inhibitors broaden the scope of analog-sensitive kinase technology. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 135, Page 18153-18159, Year 2013 |
Publish date | Aug 21, 2013 (structure data deposition date) |
Authors | Lopez, M.S. / Choy, J.W. / Peters, U. / Sos, M.L. / Morgan, D.O. / Shokat, K.M. |
External links | J. Am. Chem. Soc. / PubMed:24171479 |
Methods | X-ray diffraction |
Resolution | 2.73 Å |
Structure data | PDB-4mcv: |
Chemicals | ChemComp-29K: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase Domain / Tyrosine Kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |