| タイトル | Refined structures of mouse P-glycoprotein. |
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| ジャーナル・号・ページ | Protein Sci., Vol. 23, Page 34-46, Year 2014 |
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| 掲載日 | 2013年8月3日 (構造データの登録日) |
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著者 | Li, J. / Jaimes, K.F. / Aller, S.G. |
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リンク | Protein Sci. / PubMed:24155053 |
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| 手法 | X線回折 |
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| 解像度 | 3.8 - 4.4 Å |
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| 構造データ | PDB-4m1m: Corrected Structure of Mouse P-glycoprotein 手法: X-RAY DIFFRACTION / 解像度: 3.8 Å PDB-4m2s: Corrected Structure of Mouse P-glycoprotein bound to QZ59-RRR 手法: X-RAY DIFFRACTION / 解像度: 4.4 Å PDB-4m2t: Corrected Structure of Mouse P-glycoprotein bound to QZ59-SSS 手法: X-RAY DIFFRACTION / 解像度: 4.35 Å |
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| 化合物 | ChemComp-0JZ: (4R,11R,18R)-4,11,18-tri(propan-2-yl)-6,13,20-triselena-3,10,17,22,23,24-hexaazatetracyclo[17.2.1.1~5,8~.1~12,15~]tetracosa-1(21),5(24),7,12(23),14,19(22)-hexaene-2,9,16-trione
ChemComp-2J8: (4S,11S,18S)-4,11,18-tri(propan-2-yl)-6,13,20-triselena-3,10,17,22,23,24-hexaazatetracyclo[17.2.1.1~5,8~.1~12,15~]tetracosa-1(21),5(24),7,12(23),14,19(22)-hexaene-2,9,16-trione
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| 由来 |  mus musculus (ハツカネズミ)
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キーワード | HYDROLASE / ATP-Binding Cassette Transporter / Multidrug Efflux / Adenosine triphosphate / mercurated cysteines / Plasma membrane / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |
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