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-Structure paper
Title | Discovery of Nms-E973 as Novel, Selective and Potent Inhibitor of Heat Shock Protein 90 (Hsp90). |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 21, Page 7047-, Year 2013 |
Publish date | May 30, 2013 (structure data deposition date) |
Authors | Brasca, M.G. / Mantegani, S. / Amboldi, N. / Bindi, S. / Caronni, D. / Casale, E. / Ceccarelli, W. / Colombo, N. / De Ponti, A. / Donati, D. ...Brasca, M.G. / Mantegani, S. / Amboldi, N. / Bindi, S. / Caronni, D. / Casale, E. / Ceccarelli, W. / Colombo, N. / De Ponti, A. / Donati, D. / Ermoli, A. / Fachin, G. / Felder, E.R. / Ferguson, R.D. / Fiorelli, C. / Guanci, M. / Isacchi, A. / Pesenti, E. / Polucci, P. / Riceputi, L. / Sola, F. / Visco, C. / Zuccotto, F. / Fogliatto, G. |
External links | Bioorg. Med. Chem. / PubMed:24100158 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2 Å |
Structure data | PDB-4bqg: PDB-4bqj: |
Chemicals | ChemComp-50Q: ChemComp-HOH: ChemComp-XKL: |
Source |
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Keywords | CHAPERONE / HYDROLASE |