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-Structure paper
Title | Inhibitor selectivity between aldo-keto reductase superfamily members AKR1B10 and AKR1B1: Role of Trp112 (Trp111) |
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Journal, issue, pages | Febs Lett., Vol. 587, Page 3681-3686, Year 2013 |
Publish date | Aug 23, 2012 (structure data deposition date) |
![]() | Zhang, L. / Zhang, H. / Zhao, Y. / Li, Z. / Chen, S. / Zhai, J. / Chen, Y. / Xie, W. / Wang, Z. / Li, Q. ...Zhang, L. / Zhang, H. / Zhao, Y. / Li, Z. / Chen, S. / Zhai, J. / Chen, Y. / Xie, W. / Wang, Z. / Li, Q. / Zheng, X. / Hu, X. |
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Methods | X-ray diffraction |
Resolution | 1.92 - 2.3 Å |
Structure data | ![]() PDB-4gqg: ![]() PDB-4i5x: ![]() PDB-4jih: ![]() PDB-4jii: ![]() PDB-4jir: |
Chemicals | ![]() ChemComp-NAP: ![]() ChemComp-HOH: ![]() ChemComp-FLF: ![]() ChemComp-EPR: ![]() ChemComp-ZST: ![]() ChemComp-NA: ![]() ChemComp-SO4: |
Source |
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![]() | OXIDOREDUCTASE / alpha-beta TIM barrel / NADP-dependant oxidoreductase / NADP+ / TIM barrel / aldo-keto reductase / OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR / oxidoreductases / OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex / Structural Genomics / Structural Genomics Consortium / SGC |