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| Title | Fragment-Based Design for the Development of N-Domain Selective Angiotensin-1 Converting Enzyme Inhibitors |
|---|---|
| Journal, issue, pages | Clin. Sci., Vol. 126, Page 305-, Year 2014 |
| Publish date | Jul 12, 2013 (structure data deposition date) |
Authors | Douglas, R.G. / Sharma, R.K. / Masuyer, G. / Lubbe, L. / Zamora, I. / Acharya, K.R. / Chibale, K. / Sturrock, E.D. |
External links | Clin. Sci. / PubMed:24015848 |
| Methods | X-ray diffraction |
| Resolution | 2.2 Å |
| Structure data | ![]() PDB-4bxk: |
| Chemicals | ![]() ChemComp-PEG: ![]() ChemComp-P6G: ![]() ChemComp-1IU: ![]() ChemComp-ZN: ![]() ChemComp-CL: ![]() ChemComp-PG4: ![]() ChemComp-NAG: ![]() ChemComp-HOH: |
| Source |
|
Keywords | HYDROLASE / METALLOPROTEASE / PROTEASE INHIBITOR |
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homo sapiens (human)
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