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-Structure paper
Title | Naphthyridines as Novel Bet Family Bromodomain Inhibitors. |
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Journal, issue, pages | Chemmedchem, Vol. 9, Page 589-, Year 2014 |
Publish date | Jun 29, 2013 (structure data deposition date) |
Authors | Mirguet, O. / Lamotte, Y. / Chung, C. / Bamborough, P. / Delannee, D. / Bouillot, A. / Gellibert, F. / Krysa, G. / Lewis, A. / Witherington, J. ...Mirguet, O. / Lamotte, Y. / Chung, C. / Bamborough, P. / Delannee, D. / Bouillot, A. / Gellibert, F. / Krysa, G. / Lewis, A. / Witherington, J. / Huet, P. / Dudit, Y. / Trottet, L. / Nicodeme, E. |
External links | Chemmedchem / PubMed:24000170 |
Methods | X-ray diffraction |
Resolution | 1.4 - 1.92 Å |
Structure data | PDB-4bw1: PDB-4bw2: PDB-4bw3: PDB-4bw4: |
Chemicals | ChemComp-EDO: ChemComp-S5B: ChemComp-HOH: ChemComp-UTH: ChemComp-9BM: ChemComp-9B6: |
Source |
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Keywords | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / ANTAGONIST |