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-Structure paper
Title | Inhibitors that stabilize a closed RAF kinase domain conformation induce dimerization. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 9, Page 428-436, Year 2013 |
Publish date | Mar 25, 2013 (structure data deposition date) |
![]() | Lavoie, H. / Thevakumaran, N. / Gavory, G. / Li, J.J. / Padeganeh, A. / Guiral, S. / Duchaine, J. / Mao, D.Y. / Bouvier, M. / Sicheri, F. / Therrien, M. |
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Methods | X-ray diffraction |
Resolution | 3.09 Å |
Structure data | ![]() PDB-4jvg: |
Chemicals | ![]() ChemComp-B96: |
Source |
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![]() | Transferase/transferase inhibitor / kinase / phosphotransferase / Transferase-transferase inhibitor complex |