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-Structure paper
タイトル | Discovery of a Potent Boronic Acid Derived Inhibitor of the HCV RNA-Dependent RNA Polymerase. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 57, Page 1902-1913, Year 2014 |
掲載日 | 2013年4月22日 (構造データの登録日) |
![]() | Maynard, A. / Crosby, R.M. / Ellis, B. / Hamatake, R. / Hong, Z. / Johns, B.A. / Kahler, K.M. / Koble, C. / Leivers, A. / Leivers, M.R. ...Maynard, A. / Crosby, R.M. / Ellis, B. / Hamatake, R. / Hong, Z. / Johns, B.A. / Kahler, K.M. / Koble, C. / Leivers, A. / Leivers, M.R. / Mathis, A. / Peat, A.J. / Pouliot, J.J. / Roberts, C.D. / Samano, V. / Schmidt, R.M. / Smith, G.K. / Spaltenstein, A. / Stewart, E.L. / Thommes, P. / Turner, E.M. / Voitenleitner, C. / Walker, J.T. / Waitt, G. / Weatherhead, J. / Weaver, K. / Williams, S. / Wright, L. / Xiong, Z.Z. / Haigh, D. / Shotwell, J.B. |
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手法 | X線回折 |
解像度 | 1.7 - 2.45 Å |
構造データ | ![]() PDB-4kai: ![]() PDB-4kb7: ![]() PDB-4kbi: ![]() PDB-4ke5: ![]() PDB-4khm: ![]() PDB-4khr: |
化合物 | ![]() ChemComp-1PV: ![]() ChemComp-HOH: ![]() ChemComp-690: ![]() ChemComp-1C0: ![]() ChemComp-SO4: |
由来 |
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![]() | REPLICATION/REPLICATION INHIBITOR / HCV Polymerase / HCV NS5B / Site IV Inhibitor / boron / RNA Dependent RNA Polymerase / TRANSFERASE-TRANSFERASE INHIBITOR complex / REPLICATION-REPLICATION INHIBITOR complex / P66 / P70 / RNA directed RNA Polymerase / tar7360 / RNA-dependent RNA polymerase / Polymerase / RNA Replication / RNS Dependent RNA Polymerase |