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Title | In silico discovery of small-molecule Ras inhibitors that display antitumor activity by blocking the Ras-effector interaction. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 110, Page 8182-8187, Year 2013 |
Publish date | Aug 1, 2012 (structure data deposition date) |
Authors | Shima, F. / Yoshikawa, Y. / Ye, M. / Araki, M. / Matsumoto, S. / Liao, J. / Hu, L. / Sugimoto, T. / Ijiri, Y. / Takeda, A. ...Shima, F. / Yoshikawa, Y. / Ye, M. / Araki, M. / Matsumoto, S. / Liao, J. / Hu, L. / Sugimoto, T. / Ijiri, Y. / Takeda, A. / Nishiyama, Y. / Sato, C. / Muraoka, S. / Tamura, A. / Osoda, T. / Tsuda, K. / Miyakawa, T. / Fukunishi, H. / Shimada, J. / Kumasaka, T. / Yamamoto, M. / Kataoka, T. |
External links | Proc. Natl. Acad. Sci. USA / PubMed:23630290 |
Methods | NMR (solution) |
Structure data | PDB-2lwi: |
Chemicals | ChemComp-GNP: ChemComp-MG: ChemComp-KOB: ChemComp-HOH: |
Source |
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Keywords | SIGNALING PROTEIN/INHIBITOR / Ras / GTP-Bound Form / SIGNALING PROTEIN-INHIBITOR complex |