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-Structure paper
Title | Homopiperazine derivatives as a novel class of proteasome inhibitors with a unique mode of proteasome binding. |
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Journal, issue, pages | Plos One, Vol. 8, Page e60649-e60649, Year 2013 |
Publish date | Apr 25, 2012 (structure data deposition date) |
Authors | Kikuchi, J. / Shibayama, N. / Yamada, S. / Wada, T. / Nobuyoshi, M. / Izumi, T. / Akutsu, M. / Kano, Y. / Sugiyama, K. / Ohki, M. ...Kikuchi, J. / Shibayama, N. / Yamada, S. / Wada, T. / Nobuyoshi, M. / Izumi, T. / Akutsu, M. / Kano, Y. / Sugiyama, K. / Ohki, M. / Park, S.Y. / Furukawa, Y. |
External links | Plos One / PubMed:23593271 |
Methods | X-ray diffraction |
Resolution | 2.509 Å |
Structure data | PDB-4eu2: |
Chemicals | ChemComp-WPI: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / Proteasome inhibitor / HYDROLASE-HYDROLASE INHIBITOR complex |