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-Structure paper
Title | De novo design of protein kinase inhibitors by in silico identification of hinge region-binding fragments. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 1044-1052, Year 2013 |
Publish date | Jun 8, 2012 (structure data deposition date) |
Authors | Urich, R. / Wishart, G. / Kiczun, M. / Richters, A. / Tidten-Luksch, N. / Rauh, D. / Sherborne, B. / Wyatt, P.G. / Brenk, R. |
External links | Acs Chem. Biol. / PubMed:23534475 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-4fic: |
Chemicals | ChemComp-0UL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Hinge binding fragment / Type I / DFG-in / Tyrosine-protein kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |