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-Structure paper
Title | Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 1262-1275, Year 2013 |
Publish date | Jan 6, 2013 (structure data deposition date) |
![]() | Geurink, P.P. / van der Linden, W.A. / Mirabella, A.C. / Gallastegui, N. / de Bruin, G. / Blom, A.E. / Voges, M.J. / Mock, E.D. / Florea, B.I. / van der Marel, G.A. ...Geurink, P.P. / van der Linden, W.A. / Mirabella, A.C. / Gallastegui, N. / de Bruin, G. / Blom, A.E. / Voges, M.J. / Mock, E.D. / Florea, B.I. / van der Marel, G.A. / Driessen, C. / van der Stelt, M. / Groll, M. / Overkleeft, H.S. / Kisselev, A.F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.7 - 3.1 Å |
Structure data | ![]() PDB-4inr: ![]() PDB-4int: ![]() PDB-4inu: |
Chemicals | ![]() ChemComp-1G1: ![]() ChemComp-HOH: ![]() ChemComp-1G5: ![]() ChemComp-1G6: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / UPS / ![]() ![]() |