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-Structure paper
Title | Pyridylthiazole-based ureas as inhibitors of Rho associated protein kinases (ROCK1 and 2). |
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Journal, issue, pages | Medchemcomm, Vol. 3, Page 699-709, Year 2012 |
Publish date | Sep 19, 2011 (structure data deposition date) |
![]() | Pireddu, R. / Forinash, K.D. / Sun, N.N. / Martin, M.P. / Sung, S.S. / Alexander, B. / Zhu, J.Y. / Guida, W.C. / Schonbrunn, E. / Sebti, S.M. / Lawrence, N.J. |
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Methods | X-ray diffraction |
Resolution | 2.75 Å |
Structure data | ![]() PDB-3tv7: |
Chemicals | ![]() ChemComp-07Q: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / dimer / dimerization / myosin / TRANSFERASE-TRANSFERASE INHIBITOR complex |