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-Structure paper
Title | Activities, Crystal Structures and Molecular Dynamics of Dihydro-1H-Isoindole Derivatives, Inhibitors of HIV-1 Integrase. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 209-, Year 2013 |
Publish date | Oct 8, 2012 (structure data deposition date) |
![]() | Metifiot, M. / Maddali, K. / Johnson, B.C. / Hare, S. / Smith, S.J. / Zhao, X.Z. / Marchand, C. / Burke, T.R. / Hughes, S.H. / Cherepanov, P. / Pommier, Y. |
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Methods | X-ray diffraction |
Resolution | 2.38 - 2.85 Å |
Structure data | ![]() PDB-4bdy: ![]() PDB-4bdz: ![]() PDB-4be0: ![]() PDB-4be1: ![]() PDB-4be2: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-MG: ![]() ChemComp-CIJ: ![]() ChemComp-HOH: ![]() ChemComp-19C: ![]() ChemComp-BF3: ![]() ChemComp-NH4: ![]() ChemComp-CI4: ![]() ChemComp-XZ2: |
Source |
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![]() | TRANSFERASE/DNA / TRANSFERASE-DNA COMPLEX / PROTEIN-DNA COMPLEX / DNA INTEGRATION / ENDONUCLEASE / METAL-BINDING / MULTIFUNCTIONAL ENZYME / NUCLEASE / NUCLEOTIDYLTRANSFERASE / TRANSFERASE / VIRAL NUCLEOPROTEIN / VIRION / DNA-BINDING / ZINC BINDING / HHCC MOTIF / RECOMBINATION / INHIBITOR / RECOMBINATION-INHIBITOR-DNA COMPLEX / NUCLEUS / VIRAL PROTEIN |