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-Structure paper
Title | Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5. |
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Journal, issue, pages | Biochem. J., Vol. 449, Page 151-159, Year 2013 |
Publish date | Jun 28, 2011 (structure data deposition date) |
Authors | Senisterra, G. / Wu, H. / Allali-Hassani, A. / Wasney, G.A. / Barsyte-Lovejoy, D. / Dombrovski, L. / Dong, A. / Nguyen, K.T. / Smil, D. / Bolshan, Y. ...Senisterra, G. / Wu, H. / Allali-Hassani, A. / Wasney, G.A. / Barsyte-Lovejoy, D. / Dombrovski, L. / Dong, A. / Nguyen, K.T. / Smil, D. / Bolshan, Y. / Hajian, T. / He, H. / Seitova, A. / Chau, I. / Li, F. / Poda, G. / Couture, J.F. / Brown, P.J. / Al-Awar, R. / Schapira, M. / Arrowsmith, C.H. / Vedadi, M. |
External links | Biochem. J. / PubMed:22989411 |
Methods | X-ray diffraction |
Resolution | 1.8 - 1.82 Å |
Structure data | PDB-3smr: PDB-3ur4: |
Chemicals | ChemComp-NP7: ChemComp-EDO: ChemComp-UNX: ChemComp-HOH: ChemComp-0BW: ChemComp-CL: ChemComp-SO4: |
Source |
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Keywords | TRANSCRIPTION / WDR5 / SGC / Structural Genomics / Structural Genomics Consortium / WD repeat domain 5 / TRANSCRIPTION/INHIBITOR / TRANSCRIPTION-INHIBITOR complex |