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-Structure paper
Title | Structure-Based Discovery of Highly Selective Phosphodiesterase-9A Inhibitors and Implications for Inhibitor Design. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 8549-8558, Year 2012 |
Publish date | Aug 7, 2012 (structure data deposition date) |
Authors | Meng, F. / Hou, J. / Shao, Y.X. / Wu, P.Y. / Huang, M. / Zhu, X. / Cai, Y. / Li, Z. / Xu, J. / Liu, P. ...Meng, F. / Hou, J. / Shao, Y.X. / Wu, P.Y. / Huang, M. / Zhu, X. / Cai, Y. / Li, Z. / Xu, J. / Liu, P. / Luo, H.B. / Wan, Y. / Ke, H. |
External links | J. Med. Chem. / PubMed:22985069 |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | PDB-4gh6: |
Chemicals | ChemComp-LUO: ChemComp-ZN: ChemComp-MG: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/Hydrolase Inhibitor / PDE9A / HYDROLASE-Hydrolase Inhibitor complex |