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-Structure paper
Title | Identification of purple acid phosphatase inhibitors by fragment-based screening: promising new leads for osteoporosis therapeutics. |
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Journal, issue, pages | Chem. Biol. Drug Des., Vol. 80, Page 665-674, Year 2012 |
Publish date | Jan 29, 2012 (structure data deposition date) |
Authors | Feder, D. / Hussein, W.M. / Clayton, D.J. / Kan, M.W. / Schenk, G. / McGeary, R.P. / Guddat, L.W. |
External links | Chem. Biol. Drug Des. / PubMed:22943065 |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.7 Å |
Structure data | PDB-4dhl: PDB-4dsy: PDB-4dt2: |
Chemicals | ChemComp-ZN: ChemComp-FE: ChemComp-0K7: ChemComp-GOL: ChemComp-SO4: ChemComp-EDO: ChemComp-NAG: ChemComp-HOH: ChemComp-0LO: ChemComp-ACT: ChemComp-0LV: |
Source |
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Keywords | HYDROLASE / Catalytic C domain / N terminal domain / Phosphatase / Acid Phosphatase / Phosphoric Monoester Hydrolases / MO07123 / Maybridge / Fragment / lysosome / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |