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TitleDiscovery of diarylhydantoins as new selective androgen receptor modulators.
Journal, issue, pagesJ. Med. Chem., Vol. 55, Page 8225-8235, Year 2012
Publish dateDec 14, 2011 (structure data deposition date)
AuthorsNique, F. / Hebbe, S. / Peixoto, C. / Annoot, D. / Lefrancois, J.-M. / Duval, E. / Michoux, L. / Triballeau, N. / Lemoullec, J.M. / Mollat, P. ...Nique, F. / Hebbe, S. / Peixoto, C. / Annoot, D. / Lefrancois, J.-M. / Duval, E. / Michoux, L. / Triballeau, N. / Lemoullec, J.M. / Mollat, P. / Thauvin, M. / Prange, T. / Minet, D. / Clement-Lacroix, P. / Robin-Jagerschmidt, C. / Fleury, D. / Guedin, D. / Deprez, P.
External linksJ. Med. Chem. / PubMed:22897611
MethodsX-ray diffraction
Resolution1.7 - 1.95 Å
Structure data

PDB-3v49:
Structure of ar lbd with activator peptide and sarm inhibitor 1
Method: X-RAY DIFFRACTION / Resolution: 1.7 Å

PDB-3v4a:
Structure of ar lbd with activator peptide and sarm inhibitor 2
Method: X-RAY DIFFRACTION / Resolution: 1.95 Å

Chemicals

ChemComp-PK0:
4-[(4R)-4-(4-hydroxyphenyl)-3,4-dimethyl-2,5-dioxoimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile

ChemComp-SO4:
SULFATE ION

ChemComp-HOH:
WATER

ChemComp-PK1:
(5R)-3-(3,4-dichlorophenyl)-5-(4-hydroxyphenyl)-1,5-dimethyl-2-thioxoimidazolidin-4-one

Source
  • homo sapiens (human)
KeywordsTRANSCRIPTION / DIARYLHYDANTOIN / SYNTHESIS / SARM / ANTIANDROGEN / LIGAND BINDING DOMAIN / testosterone / Dihydrotestosterone / SARM (Selective Androgen Receptor Modulator) / ANDROGEN RECEPTOR / Selective Androgen Receptor Modulator

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