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-Structure paper
| Title | The Design, Synthesis, and Biological Evaluation of Pim Kinase Inhibitors. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 3732-, Year 2012 |
| Publish date | Mar 5, 2012 (structure data deposition date) |
Authors | Tsuhako, A.L. / Brown, D.S. / Koltun, E.S. / Aay, N. / Arcalas, A. / Chan, V. / Du, H. / Engst, S. / Franzini, M. / Galan, A. ...Tsuhako, A.L. / Brown, D.S. / Koltun, E.S. / Aay, N. / Arcalas, A. / Chan, V. / Du, H. / Engst, S. / Franzini, M. / Galan, A. / Huang, P. / Johnston, S. / Kane, B. / Kim, M.H. / Laird, A.D. / Lin, R. / Mock, L. / Ngan, I. / Pack, M. / Stott, G. / Stout, T.J. / Yu, P. / Zaharia, C. / Zhang, W. / Zhou, P. / Nuss, J.M. / Kearney, P.C. / Xu, W. |
External links | Bioorg. Med. Chem. Lett. / PubMed:22542012 |
| Methods | X-ray diffraction |
| Resolution | 1.92 - 2.6 Å |
| Structure data | ![]() PDB-4alu: ![]() PDB-4alv: ![]() PDB-4alw: |
| Chemicals | ![]() ChemComp-IMD: ![]() ChemComp-79O: ![]() ChemComp-HOH: ![]() ChemComp-R9P: ![]() ChemComp-HY7: |
| Source |
|
Keywords | TRANSFERASE / PROTO-ONCOGENE / PROTO-ONCOGENE SERINE/THREONINE-PROTEIN KINASE PIM-1 |
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homo sapiens (human)
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