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-Structure paper
Title | Identification of a Novel Family of BRAF(V600E) Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 5220-5230, Year 2012 |
Publish date | Mar 7, 2012 (structure data deposition date) |
Authors | Qin, J. / Xie, P. / Ventocilla, C. / Zhou, G. / Vultur, A. / Chen, Q. / Liu, Q. / Herlyn, M. / Winkler, J. / Marmorstein, R. |
External links | J. Med. Chem. / PubMed:22537109 |
Methods | X-ray diffraction |
Resolution | 2.55 Å |
Structure data | PDB-4e26: |
Chemicals | ChemComp-734: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / inhibitor / oncoprotein / melanoma / transferase-transferase inhibitor complex |